Reviewed by Peptide Treatments Medical Advisory Board (Medical Advisory Board)

Tesamorelin: Contraindications & Drug Interactions

Safety information for Tesamorelin including known contraindications, drug interactions, and important precautions.

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Contraindications

  • Active malignancy or history of malignancy
  • Pregnancy (Category X)
  • Disruption of hypothalamic-pituitary axis from surgery, radiation, or trauma

Drug Interactions (2 interactions)

Important: This table summarizes known and theoretical interactions. Always consult a healthcare provider before combining Tesamorelin with any medication.
Drug Classification Mechanism
Glucocorticoids Documented Corticosteroids may attenuate GH-releasing effects of tesamorelin
Insulin / oral hypoglycemics Theoretical GH elevation may increase insulin resistance

Use our interactive Drug Interaction Checker for real-time lookup.